Selective Inhibition of Bruton’s Tyrosine Kinase by a Designed Covalent Ligand Leads to Potent Therapeutic Efficacy in Blood Cancers Relative to Clinically Used Inhibitors

  1. Sousa, B.B.
  2. de Almeida, C.R.
  3. Barahona, A.F.
  4. Lopes, R.
  5. Martins-Logrado, A.
  6. Cavaco, M.
  7. Neves, V.
  8. Carvalho, L.A.R.
  9. Labaõ-Almeida, C.
  10. Coelho, A.R.
  11. Bento, M.L.
  12. Lopes, R.M.R.M.
  13. Oliveira, B.L.
  14. Castanho, M.A.R.B.
  15. Neumeister, P.
  16. Deutsch, A.
  17. Vladimer, G.I.
  18. Krall, N.
  19. Joaõ, C.
  20. Corzana, F.
  21. Seixas, J.D.
  22. Fior, R.
  23. Bernardes, G.J.L.
Journal:
ACS Pharmacology and Translational Science

ISSN: 2575-9108

Year of publication: 2022

Volume: 5

Issue: 11

Pages: 1156-1168

Type: Article

DOI: 10.1021/ACSPTSCI.2C00163 GOOGLE SCHOLAR lock_openOpen access editor
Institutional repository: lock_openOpen access Editor